多巴胺D3受体配体研究现状
The research status of dopamine D3 receptor ligands
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摘要: 综述了现有多巴胺D3受体配体(主要是氨基四氢萘满类)的分子结构、受体亲和性和受体选择性进行了比较,并对多巴胺D3受体配体的研究进行了展望。Abstract: Dopamine D3 receptor ligands were reviewed in this paper. Aminotetralin derivatives is a main kind of them. After comparing the molecule structure, receptor affinity and receptor selectivity of them, I made a prospective research future of high selective and affinity ligands of dopamine D3 receptor.
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Key words:
- dopamine /
- D3receptor /
- ligand /
- aminotetralin
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