[1] |
Currie E, Schulze A, Zechner R, et al. Cellular fatty acid metabolism and cancer[J]. Cell Metab, 2013, 18(2):153-161. DOI:10.1016/j.cmet.2013.05.017. |
[2] |
Santos CR, Schulze A. Lipid metabolism in cancer[J]. FEBS J, 2012, 279(15):2610-2623. DOI:10.1111/j.1742-4658. 2012.08644.x. |
[3] |
Gropler RJ. Recent advances in metabolic imaging[J]. J Nucl Cardiol, 2013, 20(6):1147-1172. DOI:10.1007/s12350-013-9786-z. |
[4] |
孙爱君, 任茜, 刘健, 等. 11C-乙酸盐PET和PET/CT在肿瘤显像中的应用[J].国际放射医学核医学杂志, 2013, 37(4):243-247. DOI:10.3760/cma.j.issn.1673-4114.2013.04.013. Sun AJ, Ren Q, Liu J, et al. The application of 11C-acetate PET and PET-CT for tumors[J]. Int J Radiat Med Nucl Med, 2013, 37(4):243-247. doi: 10.3760/cma.j.issn.1673-4114.2013.04.013 |
[5] |
Yoshii Y, Furukawa T, Saga T, et al. Acetate/acetyl-CoA metabolism associated with cancer fatty acid synthesis:overview and application[J]. Cancer Lett, 2015, 356(2 Pt A):211-216. DOI:10.1016/j.canlet.2014.02.019. |
[6] |
Yoshii Y, Furukawa T, Oyama N, et al. Fatty acid synthase is a key target in multiple essential tumor functions of prostate cancer:uptake of radiolabeled acetate as a predictor of the targeted therapy outcome[J/OL]. PLoS One, 2013, 8(5):e64570[2017-06-28]. http://journals.plos.org/plosone/article?id=10.1371/journal.pone.0064570. DOI:10.1371/journal.pone.0064570. |
[7] |
Zaytseva YY, Elliott VA, Rychahou P, et al. Cancer cell-associated fatty acid synthase activates endothelial cells and promotes angiogenesis in colorectal cancer[J]. Carcinogenesis, 2014, 35(6):1341-1351. DOI:10.1093/carcin/bgu042. |
[8] |
Plathow C, Weber WA. Tumor cell metabolism imaging[J]. J Nucl Med, 2008, 49 suppl 2:43S-59S. DOI:10.2967/jnumed.107. 045930. |
[9] |
Agostini M, Almeida LY, Bastos DC, et al. The fatty acid synthase inhibitor orlistat reduces the growth and metastasis of orthotopic tongue oral squamous cell carcinomas[J]. Mol Cancer Ther, 2014, 13(3):585-595. DOI:10.1158/1535-7163.MCT-12-1136. |
[10] |
Seguin F, Carvalho MA, Bastos DC, et al. The fatty acid synthase inhibitor orlistat reduces experimental metastases and angiogenesis in B16-F10 melanomas[J]. Br J Cancer, 2012, 107(6):977-987.DOI:10.1038/bjc.2012.355. |
[11] |
Brown M, Marshall DR, Sobel BE, et al. Delineation of myocardial oxygen utilization with carbon-11-labeled acetate[J]. Circulation, 1987, 76(3):687-696. DOI:10.1161/01.CIR.76.3.687. |
[12] |
Henes CG, Bergmann SR, Walsh MN, et al. Assessment of myocardial oxidative metabolic reserve with positron emission tomography and carbon-11 acetate[J]. J Nucl Med, 1989, 30(9):1489-1499. |
[13] |
Park JW, Kim JH, Kim SK, et al. A prospective evaluation of 18F-FDG and 11C-acetate PET/CT for detection of primary and metastatic hepatocellular carcinoma[J]. J Nucl Med, 2008, 49(12):1912-1921.DOI:10.2967/jnumed.108.055087. |
[14] |
Huo L, Dang Y, Lv J, et al. Application of dual phase imaging of 11C-acetate positron emission tomography on differential diagnosis of small hepatic lesions[J/OL]. PLoS One, 2014, 9(5):e96517[2016-06-28]. http://journals.plos.org/plosone/article?id=10.1371/journal.pone.0096517. DOI:10.1371/journal.pone.0096517. |
[15] |
Salem N, Kuang Y, Wang F, et al. PET imaging of hepatocellular carcinoma with 2-deoxy-2[18F] fluoro-D-glucose, 6-deoxy-6[18F]fluoro-D-glucose, [1-11C]-acetate and[N-methyl-11C]-choline[J]. Q J Nucl Med Mol Imaging, 2009, 53(2):144-156. |
[16] |
Shreve P, Chiao PC, Humes HD, et al. Carbon-11-acetate PET imaging in renal disease[J]. J Nucl Med, 1995, 36(9):1595-1601. |
[17] |
Oyama N, Okazawa H, Kusukawa N, et al. 11C-Acetate PET imaging for renal cell carcinoma[J]. Eur J Nucl Med Mol Imaging, 2009, 36(3):422-427. DOI:10.1007/s00259-008-0981-0. |
[18] |
霍力, 周前, 吴战宏, 等. 11C-乙酸盐PET显像在肾脏肿瘤诊断中的作用[J].中华核医学杂志, 2006, 26(4):205-208. DOI:10.3760/cma.j.issn.2095-2848. 2006.04.003. Huo L, Zhou Q, Wu ZH, et al. The role of 11C-acetate PET imaging for diagnosis of renal cancer[J]. Chin J Nucl Med, 2006, 26(4):205-208. doi: 10.3760/cma.j.issn.2095-2848.2006.04.003 |
[19] |
Oyama N, Akino H, Kanamaru H, et al. 11C-acetate PET imaging of prostate cancer[J]. J Nucl Med, 2002, 43(2):181-186. |
[20] |
Albrecht S, Buchegger F, Soloviev D, et al. 11C-acetate PET in the early evaluation of prostate cancer recurrence[J]. Eur J Nucl Med Mol Imaging, 2007, 34(2):185-196. DOI:10.1007/s00259-006-0163-x. |
[21] |
Brogsitter C, Zöphel K, Kotzerke J. 18F-Choline, 11C-choline and 11C-acetate PET/CT:comparative analysis for imaging prostate cancer patients[J]. Eur J Nucl Med Mol Imaging, 2013, 40 suppl 1:S18-27. DOI:10.1007/s00259-013-2358-2. |
[22] |
Tang G, Tang X, Wang M, et al. A simple and rapid automated radiosynthesis of[18F]fluoroacetate[J]. J Labelled Compd Radiopharm, 2008, 51(7):297-301. DOI:10.1002/jlcr.1520. |
[23] |
Ponde DE, Dence CS, Oyama N, et al. 18F-fluoroacetate:a potential acetate analog for prostate tumor imaging-in vivo evaluation of 18F-fluoroacetate versus 11C-acetate[J]. J Nucl Med, 2007, 48(3):420-428. |
[24] |
Lindhe O, Sun A, Ulin J, et al.[18F] Fluoroacetate is not a functional analogue of[11C]acetate in normal physiology[J]. Eur J Nucl Med Mol Imaging, 2009, 36:1453-1459. DOI:10.1007/s00259-009-1128-7. |
[25] |
Matthies A, Ezziddin S, Ulrich EM, et al. Imaging of prostate cancer metastases with 18F-fluoroacetate using PET/CT[J]. Eur J Nucl Med Mol Imaging, 2004, 31(5):797. DOI:10.1007/s00259-003-1437-1. |
[26] |
Liu RS, Chou TK, Chang CH, et al. Biodistribution, pharmacokinetics and PET imaging of[18F]FMISO, [18F]FDG and[18F]FAc in a sarcoma-and inflammation-bearing mouse model[J]. Nucl Med Biol, 2009, 36(3):305-312. DOI:10.1016/j.nucmedbio.2008.12.011. |
[27] |
周硕, 朱庆国, 叶烈夫, 等. 18F-氟乙酸联合18F-FDG PET/CT显像在肾肿瘤鉴别诊断中的价值[J].大连医科大学学报, 2016, 38(4):340-343, 360. DOI:10.11724/jdmu.2016.04.06. Zhou S, Zhu QG, Ye LF, et al. Value of 18F-flunoroacetate combined with 18F-fluorodeoxyglucose in differential diagnosis of renal masses[J]. J Dalian Med Univ, 2016, 38(4):340-343, 360. doi: 10.11724/jdmu.2016.04.06 |
[28] |
Takemoto K, Hatano E, Nishii R, et al. Assessment of[18F]-fluoroacetate PET/CT as a tumor-imaging modality:preclinical study in healthy volunteers and clinical evaluation in patients with liver tumor[J]. Ann Nucl Med, 2014, 28(4):371-380. DOI:10.1007/s12149-014-0823-z. |
[29] |
Ho CL, Cheung MK, Chen S, et al.[18F] fluoroacetate positron emission tomography for hepatocellular carcinoma and metastases:an alternative tracer for[11C] acetate?[J]. Mol Imaging, 2012, 11(3):229-239. DOI:10.2310/7290. 2011.00043. |
[30] |
Yoshimoto M, Waki A, Yonekura Y, et al. Characterization of acetate metabolism in tumor cells in relation to cell proliferation:acetate metabolism in tumor cells[J]. Nucl Med Biol, 2001, 28(2):117-122. DOI:10.1016/S0969-8051(00)00195-5. |
[31] |
Pillarsetty N, Punzalan B, Larson SM. 2-18F-Fluoropropionic acid as a PET imaging agent for prostate cancer[J]. J Nucl Med, 2009, 50(10):1709-1714. DOI:10.2967/jnumed.109.064212. |
[32] |
党永红, 蔡炯, 王玲, 等. 2-18F-氟代丙酸的自动化合成及其Micro PET肺癌小鼠显像[J].中国医学装备, 2015, 12(6):46-49. DOI:10.3969/J.ISSN.1672-8270. 2015.06.015. Dang YH, Cai J, Wang L, et al. The automated synthesis of 2-18F-fluoropropoinic acid and micro PET imaging in mice of lung cancer[J]. China Med Equip, 2015, 12(6):46-49. doi: 10.3969/J.ISSN.1672-8270.2015.06.015 |
[33] |
Wang HL, Hu KZ, Tang GH, et al. Simple and efficient automated radiosynthesis of 2-18F-fluoropropionic acid using solid-phase extraction cartridges purification[J]. J Label Compd Radiopharm, 2012, 55(2):366-370. DOI:10.1002/jlcr.2952. |
[34] |
党永红, 蔡炯, 李欣, 等. 2-18F-氟丙酸在荷乳腺癌小鼠模型中的显像性能和体内分布[J].中国医学科学院学报, 2015, 37(3):320-324. DOI:10.3881/j.issn.1000-503X.2015.03.014. Dang YH, Cai J, Li X, et al. Imaging potential and biodistribution in vivo of 2-[18F] fluoropropionic acid in breast cancer-bearing mice[J]. Acta Academiae Medicinae Sinicae, 2015, 37(3):320-324. doi: 10.3881/j.issn.1000-503X.2015.03.014 |
[35] |
Pisaneschi F, Witney TH, Iddon L, et al. Synthesis of[18F] fluoro-pivalic acid:an improved PET imaging probe for the fatty acid synthesis pathway in tumours[J]. Med Chem Commun, 2013, 4(10):1350-1353. DOI:10.1039/c3md00169e. |
[36] |
Witney TH, Pisaneschi F, Alam IS, et al. Preclinical evaluation of 3-18F-fluoro-2, 2-dimethylpropionic acid as an imaging agent for tumor detection[J]. J Nucl Med, 2014, 55(9):1506-1512. DOI:10.2967/jnumed.114.140343. |
[37] |
Brass EP. Pivalate-generating prodrugs and carnitine homeostasis in man[J]. Pharmacol Rev, 2002, 54(4):589-598. DOI:10.1124/pr.54.4.589. |